SCHEMBL10852178

SCHEMBL10852178

O=C(O)COc1ccc(Cn2ccnc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 13/20 1.00
CYP19A1 P11511 6/20 0.62
CYP11B1 P15538 1/20 0.56
CYP11B2 P19099 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10854369 0.99 TBXAS1 (1.00) TBXAS1CYP19A1
Hydrochloric Acid SCHEMBL10854125 0.97 TBXAS1 (0.97) TBXAS1CYP19A1
SCHEMBL10945811 0.87 TBXAS1 (0.78) TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL11354168 0.85 TBXAS1 (0.74) TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL10947477 0.84 TBXAS1 (0.72) TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL10849686 0.84 TBXAS1 (0.72) TBXAS1CYP19A1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL10944317 0.83 TBXAS1 (0.73) TBXAS1CYP19A1CYP11B1CYP11B2
SCHEMBL10657236 0.83 TBXAS1 (0.74) TBXAS1CYP19A1CYP11B1CYP11B2
Hydrochloric Acid SCHEMBL10751470 0.82 TBXAS1 (0.97) TBXAS1
SCHEMBL11207086 0.81 TBXAS1 (0.67) TBXAS1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4632934-A THROMBOXANE SYNTHETASE INHIBITORS KISSEI PHARMACEUTICAL CO., LTD. (JP) 1986-12-30 US disclosed
US-4555516-A FOR TREATMENT OF CARDIOVASCULAR DISORDERS PFIZER INC. (US) 1985-11-26 US disclosed
US-4448781-A CARDIOVASCULAR DISORDERS PFIZER INC. (US) 1984-05-15 US disclosed