SCHEMBL10852854

SCHEMBL10852854

O=C(NCC#CCn1ccnc1)c1ccc(Cl)cc1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.58
ALDH1A1 P00352 2/20 0.48
KDM4E B2RXH2 1/20 0.48
NPC1 O15118 1/20 0.48
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
POLB P06746 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
CYP27B1 O15528 2/20 0.47
CYP24A1 Q07973 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6571604 0.78 SMN1; SMN2 (0.84) SMN1; SMN2ALDH1A1KDM4ENPC1MAPT
SCHEMBL9029441 0.76 TBXAS1 (0.54) ALDH1A1KDM4E
SCHEMBL9715141 0.76 SMN1; SMN2 (0.77) SMN1; SMN2ALDH1A1NPC1MAPTTSHR
SCHEMBL24181493 0.73 CYP1A2 (0.54) SMN1; SMN2ALDH1A1KDM4ENPC1MAPT
SCHEMBL10247505 0.72 CYP19A1 (0.72)
Hydrochloric Acid SCHEMBL412748 0.71 CYP19A1 (0.70)
SCHEMBL6950296 0.70 TBXAS1 (0.58) SMN1; SMN2KDM4ETSHRCYP1A2CYP3A4
SCHEMBL21098369 0.70 SMN1; SMN2 (0.89) SMN1; SMN2ALDH1A1KDM4ENPC1MAPT
SCHEMBL2926364 0.70 CYP19A1 (0.78)
SCHEMBL13177000 0.69 SMN1; SMN2 (0.65) SMN1; SMN2ALDH1A1KDM4ENPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4568687-A THROMBOXANE SYNTHETASE TNZYME INHIBITORS; HYPOTENSIVE AGENTS, CARDIOTONIC AGENTS AMERICAN CYANAMID COMPANY (US) 1986-02-04 US disclosed
EP-0117462-A2 N-(2-4-(1H-imidazol-1-yl)alkyl)arylamides AMERICAN CYANAMID COMPANY (US) 1984-09-05 EP disclosed