SCHEMBL10857079

SCHEMBL10857079

CNC(=N)NC(=O)Nc1cccnc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.57
NPC1 O15118 5/20 0.57
MEN1 O00255 4/20 0.54
KMT2A Q03164 4/20 0.54
ALDH1A1 P00352 2/20 0.54
HTT P42858 2/20 0.54
KDM4E B2RXH2 2/20 0.54
LMNA P02545 3/20 0.52
MAPT P10636 3/20 0.52
CDK2 P24941 1/20 0.52
FLT4 P35916 1/20 0.52
PKM P14618 2/20 0.51
TSHR P16473 1/20 0.51
TAAR1 Q96RJ0 1/20 0.51
ATM Q13315 1/20 0.51
AHR P35869 1/20 0.50
CYP1A2 P05177 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
HIF1A Q16665 1/20 0.50
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10756618 0.88 RAB9A (0.54) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10855620 0.84 CDK2 (0.56) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10857089 0.84 RAB9A (0.54) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10857581 0.84 RAB9A (0.54) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL14538107 0.84 NPC1 (0.51) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL30633570 0.84 RAB9A (0.68) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL7785654 0.84 RAB9A (0.68) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10857086 0.82 CDK2 (0.57) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10854328 0.81 CDK2 (0.52) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10852311 0.81 CDK2 (0.52) RAB9ANPC1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed