SCHEMBL10857089

SCHEMBL10857089

CC(C)NC(=N)NC(=O)Nc1cccnc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 7/20 0.54
NPC1 O15118 7/20 0.54
MEN1 O00255 5/20 0.52
KMT2A Q03164 5/20 0.52
POLB P06746 2/20 0.51
P2RX4 Q99571 1/20 0.51
ALDH1A1 P00352 2/20 0.50
HTT P42858 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MAPT P10636 3/20 0.49
LMNA P02545 2/20 0.49
CDK2 P24941 1/20 0.49
FLT4 P35916 1/20 0.49
ATM Q13315 1/20 0.48
TSHR P16473 1/20 0.48
TAAR1 Q96RJ0 1/20 0.48
PKM P14618 2/20 0.48
FPR2 P25090 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10860771 0.87 KDM4E (0.52) RAB9ANPC1MEN1KMT2APOLB
SCHEMBL12448114 0.85 RAB9A (0.62) RAB9ANPC1MEN1KMT2APOLB
SCHEMBL10857079 0.84 RAB9A (0.57) RAB9ANPC1MEN1KMT2AALDH1A1
SCHEMBL10852311 0.83 CDK2 (0.52) RAB9ANPC1MEN1KMT2APOLB
SCHEMBL10849099 0.82 MDM2 (0.55) RAB9AMEN1KMT2AALDH1A1KDM4E
SCHEMBL10855620 0.81 CDK2 (0.56) RAB9ANPC1MEN1KMT2APOLB
SCHEMBL10857581 0.81 RAB9A (0.54) RAB9ANPC1MEN1KMT2APOLB
SCHEMBL10852749 0.80 MEN1 (0.54) RAB9ANPC1MEN1KMT2AHTT
SCHEMBL10760214 0.79 KDM4E (0.49) RAB9ANPC1MEN1KMT2APOLB
SCHEMBL10857086 0.78 CDK2 (0.57) RAB9ANPC1MEN1KMT2APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4565826-A HYPOTENSIVE, CARDIONASCULAR, ANTIULCER, ANTISECRETORY, GASTROINTESTINAL DISORDERS WILLIAM H. RORER, INC. (US) 1986-01-21 US disclosed
US-4436911-A HYPOTENSIVE, ANTISPASMODIC, ANTIULCER, ANTIPARASITIC WILLIAM H. RORER, INC. (US) 1984-03-13 US disclosed