SCHEMBL10886239

SCHEMBL10886239

COC(=O)C1=C(C)N(C(=O)c2ccco2)C(C)=CC1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
CACNA1D Q01668 4/20 0.46
ADORA3 P0DMS8 3/20 0.46
LMNA P02545 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 3/20 0.46
ABCC4 O15439 2/20 0.46
CACNA1F O60840 2/20 0.46
ABCB11 O95342 2/20 0.46
CYP1A2 P05177 2/20 0.46
ADORA2A P29274 2/20 0.46
ADORA1 P30542 2/20 0.46
OPRM1 P35372 2/20 0.46
SCN1A P35498 2/20 0.46
HTR2B P41595 2/20 0.46
KCNH2 Q12809 2/20 0.46
CACNA1S Q13698 2/20 0.46
CACNA1C Q13936 2/20 0.46
SCN5A Q14524 2/20 0.46
SCN2A Q99250 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7890630 0.84 MAPT (0.53) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL10542632 0.79 CACNA1D (0.55) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL10619732 0.77 CACNA1D (0.46) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL8405619 0.73 ADORA3 (0.44) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL7424140 0.71 ADORA3 (0.76) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL11821045 0.68 CACNA1D (0.63) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL11442155 0.68 MAPT (0.50) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL1672208 0.68 TSHR (0.70) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL9602040 0.67 CACNA1D (0.57) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2
SCHEMBL10885654 0.66 MAPT (0.73) ALDH1A1CACNA1DADORA3LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0124777-B1 1,4-DIHYDROPYRIDINE DERIVATIVES MERRELL DOW PHARMACEUTICALS INC. (US) 1986-10-29 EP disclosed