SCHEMBL10889643

SCHEMBL10889643

CSc1ccc(C(=O)C(Br)c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.48
CES1 P23141 3/20 0.48
ALDH1A1 P00352 6/20 0.47
HPGD P15428 2/20 0.47
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
PLK1 P53350 1/20 0.43
AKR1C3 P42330 1/20 0.43
AKR1C2 P52895 1/20 0.43
AKR1C1 Q04828 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
LMNA P02545 3/20 0.42
KDM4E B2RXH2 2/20 0.41
HSD17B10 Q99714 1/20 0.41
HAO1 Q9UJM8 1/20 0.40
CYP3A4 P08684 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS2R14 Q9NYV8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7845030 0.93 AKR1C3 (0.46) CES2CES1ALDH1A1HPGDMEN1
SCHEMBL4988038 0.89 PLK1 (0.42) ALDH1A1HPGDMEN1KMT2APLK1
SCHEMBL7833587 0.85 PLK1 (0.42) CES2CES1ALDH1A1HPGDMEN1
SCHEMBL6516239 0.85 PLK1 (0.42) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL7843096 0.85 PLK1 (0.42) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL28878867 0.85 ALDH1A1 (0.53) CES2CES1ALDH1A1HPGDTDP1
SCHEMBL7508723 0.84 PLK1 (0.41) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL7089429 0.84 PLK1 (0.41) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL7843939 0.84 AKR1C3 (0.48) CES2CES1ALDH1A1HPGDMEN1
SCHEMBL627867 0.82 CES2 (0.64) CES2CES1ALDH1A1TDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4576958-A VASODILATORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1986-03-18 US disclosed