SCHEMBL10901637

SCHEMBL10901637

COc1ccc2c(-c3ccncc3)occ2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 2/20 0.48
PDGFRA P16234 2/20 0.48
CYP17A1 P05093 2/20 0.44
CYP11B1 P15538 5/20 0.43
CYP11B2 P19099 5/20 0.43
NPC1 O15118 5/20 0.43
RAB9A P51151 4/20 0.43
KDM4E B2RXH2 2/20 0.42
USP2 O75604 1/20 0.42
MAPK14 Q16539 3/20 0.42
MAPK13 O15264 2/20 0.41
MAPK12 P53778 2/20 0.41
MAPK11 Q15759 2/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
CYP2D6 P10635 2/20 0.40
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 2/20 0.40
CYP19A1 P11511 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10899817 0.88 PDGFRB (0.48) PDGFRBPDGFRACYP17A1CYP11B1CYP11B2
SCHEMBL10903355 0.80 PDGFRB (0.47) PDGFRBPDGFRANPC1RAB9AKDM4E
SCHEMBL10902304 0.77 NPC1 (0.40) PDGFRBPDGFRACYP17A1NPC1RAB9A
SCHEMBL10902026 0.76 MKNK2 (0.43) PDGFRBPDGFRANPC1RAB9AKDM4E
SCHEMBL10902490 0.76 KMT2A (0.43) CYP17A1CYP11B1CYP11B2NPC1RAB9A
SCHEMBL10899791 0.76 MAPK14 (0.45) CYP17A1CYP11B1CYP11B2MAPK14MAPK13
SCHEMBL10899410 0.74 NPC1 (0.40) NPC1RAB9AKDM4EMAPK14MAPK13
SCHEMBL10901779 0.73 KIF11 (0.49) NPC1RAB9AMAPK14MAPK13MAPK12
SCHEMBL10373029 0.72 CYP2A6 (0.45) NPC1RAB9AKDM4ECYP1A2CYP3A4
SCHEMBL4514604 0.72 CYP17A1 (0.76) PDGFRBPDGFRACYP17A1CYP11B1CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4600719-A Tetrahydropyridine and piperidine derivatives CIBA GEIGY CORPORATION (US) 1986-07-15 US disclosed
US-4210655-A Anti-depressant benzofuranyl piperidines CIBA-GEIGY CORPORATION (US) 1980-07-01 US disclosed