SCHEMBL10909175

SCHEMBL10909175

Cc1cc(C(=O)Nc2c(S(=O)(=O)O)cc(O)c3ccccc23)ccc1NC(=O)C(=O)Nc1ccc(C(=O)Nc2c(S(=O)(=O)O)cc(O)c3ccccc23)cc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 2/20 0.41
DHODH Q02127 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
MEN1 O00255 5/20 0.39
KMT2A Q03164 5/20 0.39
MAPT P10636 5/20 0.39
TDP1 Q9NUW8 3/20 0.39
RAB9A P51151 3/20 0.39
LMNA P02545 2/20 0.39
CYP1A2 P05177 2/20 0.38
NPC1 O15118 2/20 0.38
MPL P40238 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KLK1 P06870 1/20 0.38
KLK5 Q9Y337 1/20 0.38
ENPP3 O14638 1/20 0.38
ENTPD3 O75355 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11348931 0.93 HPSE (0.45) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL10909512 0.91 ALDH1A1 (0.40) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL10908078 0.89 HPSE (0.44) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL10905526 0.86 DHODH (0.44) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL11438820 0.85 CASP6 (0.40) MEN1KMT2AMAPTMPLCYP2C19
SCHEMBL10907596 0.85 HPSE (0.42) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL11345247 0.84 HPSE (0.43) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL10907712 0.83 MPL (0.46) MEN1KMT2AMAPTRAB9ALMNA
SCHEMBL10907848 0.83 DHODH (0.44) HPSEDHODHTAS1R3TAS1R1TAS1R2
SCHEMBL11433569 0.83 MAPT (0.40) KMT2AMAPTTDP1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4599204-A Oxalylamides useful as dental antiplaque agents and inhibitors of connective tissue destruction AMERICAN CYANAMID COMPANY (US) 1986-07-08 US disclosed