SCHEMBL10909401

SCHEMBL10909401

CCOC(=O)CCC(NC(=O)OC(C)(C)C)c1ccccc1N

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41
CTSK P43235 5/20 0.39
TP53 P04637 1/20 0.39
CTSS P25774 1/20 0.39
NLRP3 Q96P20 1/20 0.39
MAPT P10636 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HSD17B10 Q99714 1/20 0.38
PTPRB P23467 1/20 0.38
SYK P43405 1/20 0.38
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844782 0.83 TSHR (0.50) TSHRCYP1A2CYP2C9CYP2C19HTT
SCHEMBL28499841 0.78 CTSK (0.48) TSHRCYP1A2CYP2C9CYP2C19HTT
SCHEMBL24876970 0.77 CTSK (0.47) TSHRCYP1A2CYP2C9CYP2C19HTT
SCHEMBL27387679 0.76 CTSS (0.45) CTSKCTSSMAPTALDH1A1HSD17B10
SCHEMBL6865748 0.76 ALDH1A1 (0.46) NLRP3ALDH1A1HSD17B10
SCHEMBL18683323 0.75 TSHR (0.46) TSHRCYP1A2CYP2C9CYP2C19HTT
SCHEMBL5744515 0.75 ATM (0.60) TSHRCTSKCTSSALDH1A1SYK
SCHEMBL5742902 0.75 ATM (0.60) TSHRCTSKCTSSALDH1A1SYK
SCHEMBL4596352 0.74 ATM (0.43) TSHRCTSKCTSSMAPTALDH1A1
SCHEMBL3820956 0.74 ATM (0.43) TSHRCTSKCTSSMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4575503-A ANGIOTENSIN CONVERTING ENZYME INHIBITOR, HYPOTENSIVE CIBA-GEIGY CORPORATION (US) 1986-03-11 US disclosed
US-4473575-A ANGIOTENSIN INHIBITORS, HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1984-09-25 US disclosed
US-4410520-A ANGIOTENSION CONVERTING ENZYME INGIBITOR, HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1983-10-18 US disclosed