SCHEMBL10909712

SCHEMBL10909712

CC1(Br)Cc2cc(C#N)ccc2C1=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.41
MALT1 Q9UDY8 1/20 0.39
POLB P06746 1/20 0.39
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
CYP11B2 P19099 2/20 0.36
CYP11B1 P15538 1/20 0.36
CASP3 P42574 1/20 0.36
NSD2 O96028 1/20 0.35
MAOB P27338 1/20 0.35
DRD2 P14416 2/20 0.35
DRD3 P35462 2/20 0.35
PNMT P11086 1/20 0.35
BACE1 P56817 3/20 0.33
DAO P14920 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23782830 0.78 HTR2A (0.38) PGRMALT1POLBHTR2AHTR2C
SCHEMBL10909721 0.77 METAP1 (0.42) PGRMAOBBACE1
SCHEMBL10908106 0.76 CA1 (0.41) PGRMALT1
SCHEMBL6251847 0.76 METAP1 (0.41) PGRHTR2AHTR2CHTR2BDRD2
SCHEMBL9588878 0.75 CYP11B2 (0.47) PGRMALT1HTR2AHTR2CHTR2B
SCHEMBL10341528 0.75 PGR (0.36) PGRMALT1POLBHTR2AHTR2C
SCHEMBL10341501 0.75 DGAT1 (0.42) PGRMALT1POLBMAOBALK
SCHEMBL10908361 0.72 SRD5A2 (0.46) POLB
SCHEMBL1573061 0.71 PGR (0.46) PGRMALT1POLBHTR2AHTR2C
SCHEMBL10341526 0.71 PGR (0.36) PGRMALT1POLBHTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4616013-A INOTROPIC AND VASODILATOR ACTIVITY SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-10-07 US disclosed
EP-0145236-A2 Thiadiazinone compounds, process for their preparation, and pharmaceutical compositions containing them SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1985-06-19 EP disclosed