SCHEMBL10913645

SCHEMBL10913645

CCOC(=O)Oc1cn(C2CC2)c2c(F)c(N3CCNCC3)c(F)cc2c1=O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.46
ALDH1A1 P00352 6/20 0.46
KDM4E B2RXH2 5/20 0.46
HPGD P15428 5/20 0.46
HSD17B10 Q99714 5/20 0.46
POLB P06746 2/20 0.46
OPRM1 P35372 2/20 0.46
PRKD3 O94806 1/20 0.46
ALOX15 P16050 1/20 0.46
CLK2 P49760 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
ADRB2 P07550 1/20 0.45
TOP2A P11388 3/20 0.44
TOP2B Q02880 3/20 0.44
LMNA P02545 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
PMP22 Q01453 1/20 0.43
MEN1 O00255 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10915056 0.90 KDM4E (0.50) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL9634951 0.88 ALDH1A1 (0.51) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL6776958 0.87 ADRB2 (0.59) KCNH2ALDH1A1KDM4EHPGDHSD17B10
Hydrochloric Acid SCHEMBL10501517 0.87 ALDH1A1 (0.51) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10913555 0.87 KDM4E (0.55) ALDH1A1KDM4EHPGDHSD17B10TOP2A
SCHEMBL10443823 0.86 ALDH1A1 (0.56) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10914967 0.85 ADRB2 (0.53) KCNH2ADRB2TOP2ATOP2B
SCHEMBL9677389 0.84 KCNH2 (0.53) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL10913622 0.81 ALDH1A1 (0.49) KCNH2ALDH1A1KDM4EHPGDHSD17B10
SCHEMBL7817401 0.81 ADRB2 (0.47) KCNH2ALDH1A1POLBOPRM1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0205029-A2 Quinolinecarboxylic acids with an antibacterial activity BAYER AG (DE) 1986-12-17 EP claimed
EP-0205029-A2 Quinolinecarboxylic acids with an antibacterial activity BAYER AG (DE) 1986-12-17 EP disclosed