SCHEMBL10920185

SCHEMBL10920185

O=C(O)C=CC(=O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.70
ALDH1A1 P00352 2/20 0.66
CES2 O00748 2/20 0.61
SRD5A2 P31213 1/20 0.55
LMNA P02545 2/20 0.53
P4HB P07237 1/20 0.51
KAT6A Q92794 1/20 0.50
KCNK3 O14649 1/20 0.50
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10920181 1.00 MAOB (0.70) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL11461960 0.85 MAOB (0.68) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL11461958 0.83 MAOB (0.66) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL9586253 0.83 ALDH1A1 (0.70) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL11461959 0.83 MAOB (0.66) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL977524 0.83 MAOB (1.00) MAOBALDH1A1CES2LMNAP4HB
Acetic Acid SCHEMBL10942212 0.83 MAOB (0.65) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL977523 0.83 MAOB (1.00) MAOBALDH1A1CES2LMNAP4HB
SCHEMBL29742914 0.81 CES2 (0.67) MAOBALDH1A1CES2SRD5A2LMNA
SCHEMBL1031954 0.81 CES2 (0.67) MAOBALDH1A1CES2SRD5A2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0064385-B1 2,6-DIARYL-PYRIDINECARBOXYLIC ACIDS AND THEIR THERAPEUTIC UTILITY THE UPJOHN COMPANY (US) 1986-04-02 EP disclosed
US-4377586-A Diuretic 2,6-diaryl-4-pyridine carboxylic acids THE UPJOHN COMPANY (US) 1983-03-22 US disclosed
US-4127656-A Method of inhibiting lipogensis with 3-(benzoyl)oxiranecarboxamides SHELL OIL COMPANY (US) 1978-11-28 US disclosed
US-4091221-A LIPOGENESIS INHIBITORS SHELL OIL COMPANY (US) 1978-05-23 US disclosed
US-3953463-A 2-Aryl-6-trifluoromethyl-4-pyridyl-carbinolamine antimalarials THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1976-04-27 US disclosed
US-3940404-A PLASMODIAL INFECTIONS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE ARMY (US) 1976-02-24 US disclosed