SCHEMBL10925317

SCHEMBL10925317

COc1ccc(C(N)=C(N)c2ccc(OC)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 6/20 0.67
CA2 P00918 6/20 0.67
PARP10 Q53GL7 2/20 0.67
PRSS1 P07477 1/20 0.67
PRSS2 P07478 1/20 0.67
PRSS3 P35030 1/20 0.67
PARP1 P09874 1/20 0.67
PARP2 Q9UGN5 1/20 0.67
PARP4 Q9UKK3 1/20 0.67
CES2 O00748 1/20 0.58
CES1 P23141 1/20 0.58
CA12 O43570 1/20 0.58
CA7 P43166 1/20 0.58
CA9 Q16790 1/20 0.58
CA14 Q9ULX7 1/20 0.58
ALDH1A1 P00352 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
NR1I2 O75469 1/20 0.54
PTGIR P43119 1/20 0.53
MAPK1 P28482 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29008518 0.88 CA1 (0.59) CA1CA2PARP10PRSS1PRSS2
SCHEMBL6206456 0.81 CA1 (0.62) CA1CA2PARP10PRSS1PRSS2
SCHEMBL1839900 0.81 CA1 (0.52) CA1CA2PARP10PRSS1PRSS2
SCHEMBL1839897 0.81 CA1 (0.52) CA1CA2PARP10PRSS1PRSS2
SCHEMBL201860 0.80 CA1 (0.61) CA1CA2PARP10PRSS1PRSS2
SCHEMBL428892 0.80 PRSS1 (1.00) CA1CA2PARP10PRSS1PRSS2
SCHEMBL19529679 0.80 CA1 (0.61) CA1CA2PARP10PRSS1PRSS2
SCHEMBL201761 0.80 PARP10 (1.00) CA1CA2PARP10PRSS1PRSS2
SCHEMBL1837473 0.80 CA1 (0.50) CA1CA2PARP10PRSS1PRSS2
SCHEMBL1837474 0.80 CA1 (0.50) CA1CA2PARP10PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0045081-B1 TRISUBSTITUTED IMIDAZOLE DERIVATIVES, PROCESSES FOR PREPARING THEM, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND THEIR USE CIBA-GEIGY AG (CH) 1986-01-08 EP disclosed
US-4447431-A VIRICIDES, ANTIINFLAMMATORY AND SUNCREEN AGENT CIBA-GEIGY CORPORATION (US) 1984-05-08 US disclosed
EP-0046451-A2 Diaryl-imidazole compounds, methods for their preparation, pharmaceutical drugs containing them and their use CIBA-GEIGY AG (CH) 1982-02-24 EP disclosed
EP-0045081-A2 Trisubstituted imidazole derivatives, processes for preparing them, pharmaceutical compositions containing them, and their use CIBA-GEIGY AG (CH) 1982-02-03 EP disclosed