SCHEMBL10933534

SCHEMBL10933534

C=C1C[C@@]2(CC)[C@@H](CC[C@@]2(O)C#CBr)[C@@H]2CCC3=CCCC[C@@H]3[C@@H]12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SHBG P04278 7/20 0.79
ESR1 P03372 5/20 0.79
PGR P06401 5/20 0.79
SLC6A4 P31645 5/20 0.79
AR P10275 4/20 0.79
CHRM2 P08172 3/20 0.79
SLC6A2 P23975 3/20 0.79
OPRM1 P35372 2/20 0.79
ADORA3 P0DMS8 2/20 0.79
PTGS1 P23219 2/20 0.79
SLC6A3 Q01959 2/20 0.79
NR3C1 P04150 2/20 0.79
NR1I2 O75469 2/20 0.79
DRD1 P21728 1/20 0.79
AGTR1 P30556 1/20 0.79
CCKBR P32239 1/20 0.79
DRD3 P35462 1/20 0.79
PDE4D Q08499 1/20 0.79
KCNH2 Q12809 1/20 0.79
CYP2C19 P33261 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11335079 0.91 SHBG (0.79) SHBGESR1PGRSLC6A4AR
Desogestrel SCHEMBL20353079 0.89 SHBG (1.00) SHBGESR1PGRSLC6A4AR
Desogestrel SCHEMBL41341 0.89 SHBG (1.00) SHBGESR1PGRSLC6A4AR
Desogestrel SCHEMBL14071563 0.89 SHBG (1.00) SHBGESR1PGRSLC6A4AR
Desogestrel SCHEMBL13575760 0.89 SHBG (1.00) SHBGESR1PGRSLC6A4AR
SCHEMBL16421288 0.85 PGR (0.76) SHBGESR1PGRSLC6A4AR
SCHEMBL10933347 0.84 PGR (0.80) SHBGESR1PGRSLC6A4AR
Desogestrel SCHEMBL28425701 0.84 SHBG (0.90) SHBGESR1PGRSLC6A4AR
Etonogestrel SCHEMBL14941286 0.82 SHBG (0.87) SHBGESR1PGRSLC6A4AR
SCHEMBL9619144 0.81 SHBG (0.68) SHBGESR1PGRSLC6A4AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4550100-A Process for the preparation of 17α-bromoethynyl- and 17α-iodoethynyl-17β-hydroxy steroids and novel products thereof SCHERING AKTIENGESELLSCHAFT (DE) 1985-10-29 US claimed
US-4550100-A Process for the preparation of 17α-bromoethynyl- and 17α-iodoethynyl-17β-hydroxy steroids and novel products thereof SCHERING AKTIENGESELLSCHAFT (DE) 1985-10-29 US disclosed