SCHEMBL10945003

SCHEMBL10945003

C=C(C#N)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.50
CES1 P23141 2/20 0.50
GSK3B P49841 2/20 0.47
KIF11 P52732 2/20 0.45
SRD5A2 P31213 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALOX15 P16050 1/20 0.43
BRCA1 P38398 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PTPN1 P18031 2/20 0.42
ORAI1 Q96D31 1/20 0.40
ORAI2 Q96SN7 1/20 0.40
ORAI3 Q9BRQ5 1/20 0.40
TRPV6 Q9H1D0 1/20 0.40
MGLL Q99685 1/20 0.40
DHODH Q02127 1/20 0.39
NR4A1 P22736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23621087 0.81 CES2 (0.48) CES2MEN1KMT2AALDH1A1KDM4E
SCHEMBL2979315 0.77 CES2 (0.42) CES2CES1MEN1KMT2AALDH1A1
SCHEMBL11203708 0.77 CES2 (0.59) CES2CES1GSK3BKIF11SRD5A2
SCHEMBL19114771 0.77 CES2 (0.48) CES2CES1GSK3BKIF11SRD5A2
SCHEMBL28243558 0.77 CES2 (0.58) CES2CES1GSK3BKIF11SRD5A2
SCHEMBL23389922 0.76 MAPT (0.49) MEN1KMT2AALDH1A1ALOX15HSD17B10
SCHEMBL8377031 0.75 CES2 (0.47) CES2CES1GSK3BKIF11SRD5A2
SCHEMBL4454491 0.75 MAPT (0.52) MEN1KMT2AALDH1A1KDM4EALOX15
SCHEMBL28402017 0.75 CES2 (0.56) CES2CES1GSK3BKIF11SRD5A2
SCHEMBL29056485 0.74 CES2 (0.50) CES2CES1GSK3BKIF11SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117003669-A Preparation method of unsaturated nitrile, N-15 marked unsaturated nitrile and N-15 marked rilpivirine 北京化工大学 2023-11-07 CN disclosed
US-4533655-A Analgesic dipeptide amides and method of use and compositions thereof STERLING DRUG INC. (US) 1985-08-06 US disclosed