SCHEMBL1095460

SCHEMBL1095460

N#CC(CO)c1cc(Cl)ccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
TSHR P16473 3/20 0.36
HSD17B10 Q99714 2/20 0.36
CYP3A4 P08684 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
MAPT P10636 1/20 0.36
GAA P10253 1/20 0.36
TP53 P04637 4/20 0.35
GABRA1 P14867 4/20 0.34
GABRG2 P18507 4/20 0.34
GABRB3 P28472 4/20 0.34
GABRB1 P18505 2/20 0.34
GABRB2 P47870 2/20 0.34
CCR1 P32246 1/20 0.34
CRHR1 P34998 1/20 0.33
POLB P06746 2/20 0.33
LMNA P02545 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1095213 0.86 ALDH1A1 (0.45) ALDH1A1TSHRHSD17B10MAPTGAA
SCHEMBL1095890 0.79 ESR1 (0.48) ALDH1A1TSHRCYP3A4MAPTGAA
SCHEMBL1096025 0.78 CCR1 (0.43) ALDH1A1TSHRCYP3A4TDP1MAPT
SCHEMBL1096665 0.77 KMT2A (0.38) TSHRHSD17B10TDP1MAPTGAA
SCHEMBL1095274 0.77 LMNA (0.34) TSHRTDP1MAPTGAATP53
SCHEMBL17755061 0.76 TP53 (0.42) ALDH1A1TSHRHSD17B10CYP3A4TDP1
SCHEMBL1096585 0.76 USP2 (0.41) ALDH1A1GAAGABRA1GABRG2GABRB3
SCHEMBL1096024 0.74 LMNA (0.34) ALDH1A1TDP1MAPTGAACCR1
SCHEMBL1094322 0.73 ESR1 (0.44) ALDH1A1TSHRCYP3A4TDP1MAPT
SCHEMBL8134898 0.73 TP53 (0.41) ALDH1A1TSHRHSD17B10CYP3A4TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2148854-B1 ESTERS OF 2-PHENYLALKANENITRILES AND ANTIFUNGAL COMPOSITIONS CONTAINING THEM STOUTAMIRE DONALD WESLEY (US) 2013-02-20 EP disclosed
US-8153688-B2 Esters of 2-phenylalkanenitriles and antifungal compositions containing them MCS Laboratories, Inc. (US) 2012-04-10 US disclosed
EP-2148854-A2 ESTERS OF 2-PHENYLALKANENITRILES AND ANTIFUNGAL COMPOSITIONS CONTAINING THEM Stoutamire, Donald Wesley (US) 2010-02-03 EP disclosed
US-20100022640-A1 ESTERS OF 2-PHENYLALKANENITRILES AND ANTIFUNGAL COMPOSITIONS CONTAINING THEM MCS LABORATORIES INC. 2010-01-28 US disclosed
US-7622504-B2 Esters of 2-phenylalkanenitriles and antifungal compositions containing them MCS Laboratories, Inc. (US) 2009-11-24 US disclosed
WO-2008088538-A2 ESTERS OF 2-PHENYLALKANENITRILES AND ANTIFUNGAL COMPOSITIONS CONTAINING THEM STOUTAMIRE DONALD WESLEY (US) 2008-07-24 WO disclosed
US-20080153905-A1 Esters of 2-phenylalkanenitriles and antifungal compositions containing them MCS LABORATORIES INC. 2008-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100022640-A1 ESTERS OF 2-PHENYLALKANENITRILES AND ANTIFUNGAL COMPOSITIONS CONTAINING THEM CYP51A1, ERG28, AKR7A2 ALDH1A1 1232/4885TSHR 4784/4885HSD17B10 603/4885
US-20080153905-A1 Esters of 2-phenylalkanenitriles and antifungal compositions containing them CYP51A1, ERG28, AKR7A2 ALDH1A1 1232/4885TSHR 4784/4885HSD17B10 603/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.