SCHEMBL10964644

SCHEMBL10964644

N#Cc1ccc(-c2ccc(-c3cccs3)cn2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.47
CHEK1 O14757 1/20 0.43
GAA P10253 1/20 0.43
KDM4E B2RXH2 6/20 0.42
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.42
CYP11B1 P15538 1/20 0.42
HPGD P15428 2/20 0.42
HTT P42858 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CYP2E1 P05181 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
MAPT P10636 3/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10964561 0.98 KDM1A (0.46) KDM1ACHEK1GAAKDM4EALDH1A1
SCHEMBL10727341 0.85 CHEK1 (0.41) CHEK1GAAKDM4EALDH1A1LMNA
SCHEMBL4344657 0.83 LTA4H (0.52) GAAKDM4EALDH1A1LMNACYP11B1
SCHEMBL1461854 0.82 MEN1 (0.47) GAAKDM4EALDH1A1LMNACYP11B1
SCHEMBL10160337 0.82 KDM4E (0.55) GAAKDM4EALDH1A1CYP11B1HPGD
SCHEMBL7449452 0.81 LTA4H (0.50) GAAKDM4EALDH1A1LMNACYP11B1
SCHEMBL13917342 0.81 CYP2C9 (0.53) CHEK1GAAKDM4EALDH1A1CYP11B1
SCHEMBL9021143 0.81 KDM1A (0.58) KDM1AGAAKDM4EALDH1A1CYP11B1
SCHEMBL10408880 0.79 KDM4E (0.52) GAAKDM4EALDH1A1CYP11B1HPGD
SCHEMBL10726997 0.79 FYN (0.58) KDM1ACHEK1KDM4EALDH1A1CYP2E1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0146862-A2 Pyridyl thiophenes MERCK PATENT GmbH (DE) 1985-07-03 EP disclosed