SCHEMBL10967158

SCHEMBL10967158

CC(C)Nc1nc2c(s1)CCc1[nH]c(=O)ccc1-2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
XIAP P98170 1/20 0.39
GRM4 Q14833 10/20 0.39
ALOX5 P09917 1/20 0.38
POLB P06746 1/20 0.38
KCNH2 Q12809 1/20 0.36
MAPT P10636 4/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
TP53 P04637 2/20 0.35
NPY5R Q15761 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10933747 0.63 NPY5R (0.37) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL4159209 0.62 ALDH1A1 (0.39) XIAPMAPTKDM4EALDH1A1
SCHEMBL12890455 0.59 TSHR (0.54) POLBMAPTSMN1; SMN2TP53KDM4E
SCHEMBL13482127 0.58 PKN1 (0.44) POLBMAPTSMN1; SMN2KDM4EALDH1A1
SCHEMBL866759 0.58 PKN1 (0.47) POLBMAPTMEN1ALDH1A1KMT2A
SCHEMBL10856741 0.57 SHMT2 (0.39) XIAPALOX5MAPTKDM4EMEN1
SCHEMBL21146034 0.57 PDCD1 (0.39) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL31252938 0.56 MEN1 (0.45) POLBSMN1; SMN2KDM4EMEN1ALDH1A1
SCHEMBL9994867 0.56 GRM4 (0.82) GRM4KCNH2
SCHEMBL5902421 0.55 CA12 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154190-A1 Pyridones MERCK PATENT GmbH (DE) 1985-09-11 EP disclosed