SCHEMBL10967338

SCHEMBL10967338

CN(C)C(=O)c1cccc2c1C(=O)NC2=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.59
KDM4E B2RXH2 5/20 0.50
ALDH1A1 P00352 4/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 2/20 0.50
GAA P10253 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CASP3 P42574 5/20 0.44
POLB P06746 2/20 0.42
RXFP1 Q9HBX9 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
GSK3B P49841 2/20 0.41
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
LIG1 P18858 1/20 0.39
PARP1 P09874 1/20 0.39
GSK3A P49840 1/20 0.38
CDK5 Q00535 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5128860 0.81 KDM4E (0.58) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10963820 0.80 TP53 (0.57) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL11017212 0.80 KDM4E (0.42) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL11021464 0.79 KEAP1 (0.42) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL439731 0.79 LIG1 (0.56) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL10339858 0.77 KEAP1 (0.56) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL2424940 0.77 KDM4E (0.54) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL11358929 0.77 KDM4E (0.54) KDM4EALDH1A1HPGDHSD17B10GAA
SCHEMBL11022685 0.76 KDM4E (0.39) KEAP1KDM4EALDH1A1HPGDHSD17B10
SCHEMBL11017927 0.76 KDM4E (0.41) KEAP1KDM4EALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106133984-A Addition agent of non-aqueous electrolyte, nonaqueous electrolytic solution and electrical storage device 住友精化株式会社 2016-11-16 CN disclosed
US-4556651-A Secalonic acid derivatives as antitumor agents ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1985-12-03 US disclosed
EP-0064199-B1 NOVEL SECALONIC ACID DERIVATIVES AND METHOD FOR PREPARING THEREOF Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1985-08-21 EP disclosed
US-4418061-A ANTITUMOR AGENTS ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1983-11-29 US disclosed
EP-0064199-A1 Novel secalonic acid derivatives and method for preparing thereof Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-11-10 EP disclosed