SCHEMBL10969403

SCHEMBL10969403

O=C(O)[C@]1(SCc2ccccc2)CCCN1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
CYP2C19 P33261 2/20 0.36
HRH3 Q9Y5N1 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
AKR1C1 Q04828 1/20 0.34
IDO1 P14902 3/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5698070 0.82 HTR2C (0.41) HRH3SMN1; SMN2KMT2AALDH1A1CYP3A4
SCHEMBL642483 0.76 AKR1C1 (0.37) SLC6A2SLC6A4SLC6A3AKR1C1MEN1
SCHEMBL7364415 0.76 AKR1C1 (0.37) SLC6A2SLC6A4SLC6A3AKR1C1MEN1
Bromide SCHEMBL7340605 0.75 AKR1C1 (0.36) SLC6A2SLC6A4SLC6A3AKR1C1MEN1
Hydrochloric Acid SCHEMBL1357987 0.75 AKR1C1 (0.36) SLC6A2SLC6A4SLC6A3AKR1C1MEN1
SCHEMBL9297313 0.74 ARG1 (0.35)
SCHEMBL18280876 0.74 ARG1 (0.35) CYP2C19L3MBTL1
SCHEMBL7339201 0.74 ARG1 (0.35)
SCHEMBL7339204 0.74 ARG1 (0.35)
SCHEMBL18280875 0.73 AKR1C1 (0.34) SLC6A2SLC6A4SLC6A3CYP2C19AKR1C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160355802-A1 Compositions and Methods Of Use Thereof For Making Polypeptides With Many Instances Of Nonstandard Amino Acids YALE UNIVERSITY 2016-12-08 US disclosed
EP-0053902-B1 PHOSPHINYLALKANOYL SUBSTITUTED PROLINES E.R. Squibb & Sons, Inc. (US) 1985-04-03 EP disclosed
US-4462943-A HYPOTENSIVE AGENTS E. R. SQUIBB & SONS, INC. (US) 1984-07-31 US disclosed
EP-0053902-A1 Phosphinylalkanoyl substituted prolines E.R. Squibb & Sons, Inc. (US) 1982-06-16 EP disclosed
EP-0052991-A1 Carboxyalkyl amino acid derivatives of various substituted prolines E.R. Squibb & Sons, Inc. (US) 1982-06-02 EP disclosed