SCHEMBL7364415

SCHEMBL7364415

O=C(O)[C@@]1(Sc2ccccc2)CCCN1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C1 Q04828 1/20 0.37
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
NPSR1 Q6W5P4 2/20 0.33
HSD11B1 P28845 2/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
SLC22A12 Q96S37 3/20 0.32
FFAR1 O14842 1/20 0.32
GRM5 P41594 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
MAPT P10636 2/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
NAMPT P43490 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
PLIN1 O60240 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL642483 1.00 AKR1C1 (0.37) AKR1C1SLC6A2SLC6A4SLC6A3NPSR1
Hydrochloric Acid SCHEMBL1357987 0.98 AKR1C1 (0.36) AKR1C1SLC6A2SLC6A4SLC6A3NPSR1
Bromide SCHEMBL7340605 0.98 AKR1C1 (0.36) AKR1C1SLC6A2SLC6A4SLC6A3NPSR1
Bromide SCHEMBL7342624 0.84 EPHX1 (0.38) SLC6A2SLC6A4SLC6A3ALDH1A1HPGD
Bromide SCHEMBL7347333 0.79 ELANE (0.40) SLC6A2SLC6A3NPSR1ALDH1A1HPGD
SCHEMBL7366551 0.78 OPRM1 (0.32)
SCHEMBL10969403 0.76 SLC6A2 (0.37) AKR1C1SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL18280875 0.76 AKR1C1 (0.34) AKR1C1SLC6A2SLC6A4SLC6A3NPSR1
SCHEMBL7380300 0.76 ELANE (0.31)
SCHEMBL11234892 0.72 ALDH1A1 (0.39) AKR1C1ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4736066-A Intermediate for substituted peptide compounds E. R. SQUIBB & SONS, INC. (US) 1988-04-05 US disclosed
US-4535176-A HYPOTENSIVE AGENTS, ANALGESICS, ANGIOTENSIN CONVERTING ENZYME INHIBITORS E. R. SQUIBB & SONS, INC. (US) 1985-08-13 US disclosed
US-4514391-A HYPOTENSIVE AGENTS; ANALGESICS E. R. SQUIBB & SONS, INC. (US) 1985-04-30 US disclosed
EP-0132304-A2 Hydroxy substituted peptide compounds E.R. Squibb & Sons, Inc. (US) 1985-01-30 EP disclosed
US-4470973-A HYPOTENSIVE AGENTS, ANALGESICS E. R. SQUIBB & SONS, INC. (US) 1984-09-11 US disclosed