SCHEMBL10969876

SCHEMBL10969876

Cc1sc(C(=O)CCc2ccccc2)c(O)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
SLC5A1 P13866 1/20 0.46
SLC5A2 P31639 1/20 0.46
KEAP1 Q14145 1/20 0.46
CYP1A1 P04798 1/20 0.46
CYP1B1 Q16678 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
FFAR1 O14842 1/20 0.43
TDP1 Q9NUW8 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RECQL P46063 2/20 0.43
HTT P42858 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALOX5 P09917 1/20 0.42
POLB P06746 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1844262 0.76 SLC5A1 (0.58) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL9808385 0.75 ALDH1A1 (0.47) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL11239913 0.75 SLC5A1 (0.54) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL11526781 0.71 NPC1 (0.56) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL457057 0.71 SLC5A1 (0.65) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL10971703 0.69 GAA (0.54) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL12330301 0.68 NPC1 (0.70) ALDH1A1MAPTKEAP1NPC1RAB9A
SCHEMBL27889179 0.68 RECQL (0.62) ALDH1A1KEAP1CYP1A1CYP1B1NPC1
SCHEMBL30572 0.68 TDP1 (0.77) ALDH1A1GAAMAPTSLC5A1SLC5A2
SCHEMBL15524969 0.68 TDP1 (0.77) ALDH1A1GAAMAPTSLC5A1SLC5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0053603-B1 1-(3-(2-HYDROXY-3-ALKYLAMINOPROPOXY)-2-THIENYL)-3-PHENYL-1 PROPANONES AND THEIR ACID ADDITION SALTS, AND PROCESS FOR THEIR PREPARATION Laevosan-Gesellschaft m.b.H. & Co KG (AT) 1985-04-03 EP disclosed
US-4352819-A ANTIARRHYTHMIA AGENTS LAEVOSAN-GESELLSCHAFT MBH & CO. KG (AT) 1982-10-05 US disclosed