SCHEMBL10970599

SCHEMBL10970599

CCCCC(=O)OCC.COc1cc2[nH]c(=O)nc(C)c2cc1OC

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TNF P01375 16/20 0.50
PDE3B Q13370 1/20 0.46
PDE3A Q14432 1/20 0.46
GABRA1 P14867 2/20 0.46
GABRA5 P31644 2/20 0.46
GABRA3 P34903 2/20 0.46
GABRA2 P47869 2/20 0.46
GABRA6 Q16445 2/20 0.46
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
HPGD P15428 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
GABRG2 P18507 1/20 0.42
GABRB3 P28472 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10974105 0.94 GABRA1 (0.48) TNFPDE3BPDE3AGABRA1GABRA5
SCHEMBL7408010 0.81 PDE3B (0.60) PDE3BPDE3AGABRA1GABRA5GABRA3
SCHEMBL11116678 0.78 PDE3B (0.51) PDE3BPDE3AGABRA1GABRA5GABRA3
Valeric Acid SCHEMBL10968822 0.72 GPR35 (0.38) KDM4EALDH1A1HPGD
SCHEMBL10974103 0.70 TNF (0.61) TNFGAA
SCHEMBL10970598 0.70 TNF (0.57) TNF
SCHEMBL7414959 0.69 PDE3B (0.56) PDE3BPDE3AGABRA1GABRA5GABRA3
SCHEMBL10985135 0.68 TNF (0.54) TNFALDH1A1HPGD
SCHEMBL11045667 0.66 CYP1A2 (0.61) ALDH1A1GAA
SCHEMBL127083 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4556739-A QUINAZOLINONE INTERMEDIATES ORTHO PHARMACEUTICAL CORPORATION (US) 1985-12-03 US disclosed
EP-0138492-A2 Process for preparing substituted 4-alkyl-2(1H) quinazolinone-1-alkanoic acid derivatives ORTHO PHARMACEUTICAL CORPORATION (US) 1985-04-24 EP disclosed