SCHEMBL10972136

SCHEMBL10972136

[O-][S+]1CCN(c2nc(Cl)nc3c(NCCCCc4ccccc4)ncnc23)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADK P55263 3/20 0.42
ADORA1 P30542 5/20 0.40
ADORA3 P0DMS8 3/20 0.40
MAPT P10636 1/20 0.40
ADORA2A P29274 4/20 0.39
TMIGD3 P0DMS9 2/20 0.39
ABCC1 P33527 2/20 0.39
ABCG2 Q9UNQ0 2/20 0.39
ADORA2B P29275 1/20 0.39
ABCB1 P08183 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3R1 P27986 1/20 0.39
TSHR P16473 2/20 0.39
LMNA P02545 1/20 0.39
HSD17B10 Q99714 1/20 0.39
HUWE1 Q7Z6Z7 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10664114 0.97 ADK (0.43) ADKADORA1ADORA3MAPTADORA2A
SCHEMBL10660880 0.93 NPSR1 (0.43) ADKADORA1MAPTADORA2ATMIGD3
SCHEMBL10663431 0.87 PDE4A (0.48) ADORA1ADORA2ATMIGD3ADORA2BLMNA
SCHEMBL11062725 0.86 PDE4A (0.43) ADKADORA1ADORA3ADORA2ATMIGD3
SCHEMBL10661153 0.86 PDE5A (0.38) MAPTLMNAPOLB
SCHEMBL11049123 0.85 PDE5A (0.39) MAPTLMNAPOLB
SCHEMBL10658083 0.84 KHK (0.42) LMNAHSD17B10NPSR1POLB
SCHEMBL10662680 0.84 CCNB2 (0.38) TSHRLMNAHSD17B10NPSR1PDE4A
SCHEMBL10970652 0.83 HRH4 (0.44) ABCC1ABCG2ABCB1TSHRPDE4A
SCHEMBL8851152 0.83 ADK (0.55) ADKADORA1ADORA3MAPTADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055444-B1 TRISUBSTITUTED PYRIMIDO(5,4-D)PYRIMIDINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1985-03-20 EP disclosed
US-4478833-A ANTICOAGULANTS DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-10-23 US disclosed
EP-0055444-A2 Trisubstituted pyrimido(5,4-d)pyrimidines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-07-07 EP disclosed