SCHEMBL8851152

SCHEMBL8851152

Clc1nc(N2CCOCC2)c2ncnc(NCCCc3ccccc3)c2n1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADK P55263 4/20 0.55
ALDH1A1 P00352 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PIK3CD O00329 1/20 0.43
PIK3R1 P27986 1/20 0.43
OGA O60502 1/20 0.43
ADORA2A P29274 4/20 0.43
ADORA1 P30542 4/20 0.43
TMIGD3 P0DMS9 3/20 0.43
ABCC1 P33527 2/20 0.43
ABCG2 Q9UNQ0 2/20 0.43
ADORA2B P29275 2/20 0.43
ABCB1 P08183 1/20 0.43
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
ACHE P22303 1/20 0.43
GAA P10253 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8851160 0.94 ADK (0.54) ADKALDH1A1MEN1KMT2AOGA
SCHEMBL8851335 0.88 PDE4A (0.55) ALDH1A1PDE4APDE4BPDE4CPDE4D
SCHEMBL10664114 0.86 ADK (0.43) ADKPIK3CDPIK3R1ADORA2AADORA1
SCHEMBL10972136 0.83 ADK (0.42) ADKPIK3CDPIK3R1ADORA2AADORA1
SCHEMBL11047372 0.82 ACHE (0.49) ADKALDH1A1ADORA2AADORA1TMIGD3
SCHEMBL9232181 0.80 ADK (0.48) ADKPIK3CDADORA2AADORA1TMIGD3
SCHEMBL10660880 0.80 NPSR1 (0.43) ADKALDH1A1ADORA2AADORA1TMIGD3
SCHEMBL10663616 0.80 ALDH1A1 (0.43) ADKALDH1A1OGAPDE4APDE4B
SCHEMBL10664729 0.80 ADORA2A (0.53) ALDH1A1MEN1KMT2AADORA2AMAPT
SCHEMBL11028726 0.79 OGA (0.53) ADKALDH1A1MEN1KMT2APIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618814-A Trisubstituted pyrimido [5,4-d] pyrimidines for modulating multi-drug resistance and pharmaceutical compositions containing these compounds DR. KARL THOMAE GMBH (DE) 1997-04-08 US disclosed
EP-0645390-A1 Trisubstituted pyrimido 5,4-d pyrimidines for modulating multidrug resistance, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1995-03-29 EP disclosed