SCHEMBL10979014

SCHEMBL10979014

O=C(Cc1ncc(Br)c(=S)[nH]1)c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
RAB9A P51151 4/20 0.43
MAPT P10636 4/20 0.43
SMN1; SMN2 Q16637 4/20 0.43
GSK3B P49841 2/20 0.39
PTPN1 P18031 1/20 0.39
KDM6B O15054 1/20 0.39
KDM4A O75164 1/20 0.39
KDM4D Q6B0I6 1/20 0.39
KDM3B Q7LBC6 1/20 0.39
HIF1AN Q9NWT6 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
KDM2A Q9Y2K7 1/20 0.39
NPC1 O15118 4/20 0.38
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 4/20 0.38
GLA P06280 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10974338 0.81 MAPT (0.41) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
SCHEMBL5523498 0.76 NPC1 (0.47) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
Hydrochloric Acid SCHEMBL5850214 0.75 RAB9A (0.46) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
SCHEMBL10986706 0.71 CTNNB1 (0.44) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
Bromide SCHEMBL10981550 0.70 CTNNB1 (0.43) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
SCHEMBL5849864 0.67 RAB9A (0.47) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
SCHEMBL4968860 0.66 GAA (0.61) ALDH1A1RAB9AMAPTSMN1; SMN2NPC1
SCHEMBL31158393 0.65 ADORA3 (0.49) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B
Hydrochloric Acid SCHEMBL5851393 0.65 GAA (0.59) ALDH1A1MAPTSMN1; SMN2KMT2AMEN1
SCHEMBL2936987 0.64 GSK3B (0.52) ALDH1A1RAB9AMAPTSMN1; SMN2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0033195-B1 PYRIMIDINE-2-SULPHIDES AND THEIR S-OXIDES FOR USE IN MEDICINE, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, PROCESSES FOR THEIR PREPARATION AND SUCH COMPOUNDS WHEN NOVEL PER SE NYEGAARD & CO. A/S (NO) 1985-12-04 EP disclosed
US-4423047-A INHIBITING ABNORMAL CELL PROLIFERATION NYEGAARD & CO. A/S (NO) 1983-12-27 US disclosed
EP-0033195-A1 Pyrimidine-2-sulphides and their S-oxides for use in medicine, pharmaceutical compositions containing them, processes for their preparation and such compounds when novel per se NYEGAARD & CO. A/S (NO) 1981-08-05 EP disclosed