Phosphoramidic Acid

Phosphoramidic Acid

SCHEMBL109796

NP(=O)(O)O.Nc1nc2c(ncn2[C@@H]2O[C@H](C(O)N(CCCC(=O)O)CCCC(=O)O)[C@@H](O)[C@H]2O)c(=O)[nH]1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NT5E P21589 1/20 0.52
HINT1 P49773 5/20 0.50
TGM2 P21980 1/20 0.49
TAAR1 Q96RJ0 1/20 0.49
HPRT1 P00492 1/20 0.48
KRAS P01116 6/20 0.47
GSK3A P49840 2/20 0.46
RPS6KA3 P51812 2/20 0.46
MAPK14 Q16539 2/20 0.46
IMPDH2 P12268 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phosphoramidic Acid SCHEMBL112033 0.96 NT5E (0.53) NT5EHINT1TGM2TAAR1HPRT1
Phosphoramidic Acid SCHEMBL108470 0.91 NT5E (0.54) NT5EHINT1TGM2TAAR1KRAS
Phosphoramidic Acid SCHEMBL111677 0.86 POLB (0.52) NT5EHPRT1
Phosphoramidic Acid SCHEMBL111868 0.84 GNMT (0.56) NT5E
Phosphoramidic Acid SCHEMBL112292 0.82 POLB (0.53) NT5ETGM2TAAR1HPRT1KRAS
SCHEMBL22636005 0.80 NT5E (0.62) NT5EHINT1TGM2TAAR1KRAS
SCHEMBL22498538 0.80 NT5E (0.62) NT5EHINT1TGM2TAAR1KRAS
SCHEMBL7535718 0.79 HINT1 (0.58) NT5EHINT1TGM2TAAR1KRAS
Phosphoramidic Acid SCHEMBL109493 0.79 QARS1 (0.56)
SCHEMBL11163143 0.79 HINT1 (0.58) NT5EHINT1TGM2TAAR1KRAS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120108533-A1 NOVEL PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U.LEUVEN R&D (BE) 2012-05-03 US disclosed
EP-2424874-A1 NOVEL PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL ANGENTS Katholieke Universiteit Leuven, K.U. Leuven R&D (BE) 2012-03-07 EP disclosed
WO-2010125200-A1 NOVEL PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL ANGENTS KATHOLIEKE UNIVERSITEIT LEUVEN, K.U. LEUVEN R&D (BE) 2010-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120108533-A1 NOVEL PHOSPHATE MODIFIED NUCLEOSIDES USEFUL AS SUBSTRATES FOR POLYMERASES AND AS ANTIVIRAL AGENTS PNP, TYMP, MTAP NT5E 253/4885HINT1 119/4885TGM2 4080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.