SCHEMBL10988515

SCHEMBL10988515

COc1cc2c(c(C)c1Cl)OCC(C(O)CN1CCNCC1)O2

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 1/20 0.36
CD274 Q9NZQ7 1/20 0.36
ALDH1A1 P00352 1/20 0.33
HTR4 Q13639 1/20 0.32
IDO1 P14902 1/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
CYP1A2 P05177 1/20 0.30
CHRM2 P08172 1/20 0.30
SLC6A4 P31645 1/20 0.30
OPRD1 P41143 1/20 0.30
OPRK1 P41145 1/20 0.30
SLC6A2 P23975 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7446683 0.82 HTR1A (0.32)
SCHEMBL10992158 0.82 IDO1 (0.33) IDO1
SCHEMBL7431643 0.82 HTR4 (0.32) HTR4
SCHEMBL10993826 0.81 BACE1 (0.32) SLC6A4SLC6A2
SCHEMBL10996604 0.76 SIGMAR1 (0.35) SLC6A4SLC6A2
SCHEMBL10992177 0.76 SMN1; SMN2 (0.35) ALDH1A1IDO1
SCHEMBL10992228 0.75 SLC6A2 (0.40) ALDH1A1HTR3EHTR3BHTR3AHTR3D
SCHEMBL10992659 0.73 SLC6A2 (0.37) CYP1A2SLC6A4SLC6A2
SCHEMBL10991101 0.73 SLC6A2 (0.37) CYP1A2SLC6A4SLC6A2
SCHEMBL10989799 0.73 IDO1 (0.34) ALDH1A1IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed