SCHEMBL10993277

SCHEMBL10993277

CS(=O)(=O)c1ccc2c(c1)OCC(C(O)CN1CCN(CC(=O)Nc3cc(F)cc(F)c3)CC1)O2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
KMT2A Q03164 3/20 0.45
CYP1A2 P05177 3/20 0.45
CYP3A4 P08684 3/20 0.45
CYP2D6 P10635 3/20 0.45
CYP2C19 P33261 3/20 0.45
CYP2C9 P11712 2/20 0.45
MEN1 O00255 2/20 0.45
TSHR P16473 4/20 0.43
GAA P10253 2/20 0.42
MAPK1 P28482 1/20 0.42
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
CA7 P43166 3/20 0.42
POLB P06746 1/20 0.42
CHRNB2 P17787 2/20 0.40
CHRNB4 P30926 2/20 0.40
CHRNA3 P32297 2/20 0.40
CHRNA4 P43681 2/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7439355 0.88 ALDH1A1 (0.41) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL10996565 0.86 TSHR (0.46) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL10997355 0.86 POLB (0.55) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL10993275 0.81 FFAR1 (0.34) CYP3A4CYP2D6CA1CA2CA7
SCHEMBL10995111 0.80 LMNA (0.50) ALDH1A1KMT2AMEN1TSHRGAA
SCHEMBL10994694 0.78 AKR1B1 (0.36) ALDH1A1CA1CA2POLBLMNA
SCHEMBL10995044 0.77 ALDH1A1 (0.48) ALDH1A1KMT2AMEN1GAAPOLB
SCHEMBL10993684 0.77 ALDH1A1 (0.48) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL10991656 0.77 ALDH1A1 (0.61) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL10994397 0.76 ALDH1A1 (0.58) ALDH1A1KMT2ACYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed