SCHEMBL10996291

SCHEMBL10996291

CN(C)CCC(Oc1cccc(C(F)(F)F)c1)C1CC1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.44
SLC6A4 P31645 2/20 0.43
HRH3 Q9Y5N1 1/20 0.43
PPARG P37231 4/20 0.41
KDM4E B2RXH2 2/20 0.41
PPARA Q07869 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40
FFAR1 O14842 2/20 0.39
GAA P10253 2/20 0.38
UTS2R Q9UKP6 1/20 0.38
HPGD P15428 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10985607 0.85 ALDH1A1 (0.58) SLC6A9PPARGKDM4EPPARAALDH1A1
SCHEMBL10989251 0.84 SLC6A4 (0.56) SLC6A9SLC6A4HRH3KDM4ESLC6A2
SCHEMBL10985198 0.83 TAAR1 (0.41) SLC6A4PPARGPPARASLC6A2SLC6A3
SCHEMBL10989204 0.82 SLC6A4 (0.46) SLC6A4HRH3PPARGKDM4EPPARA
SCHEMBL10995397 0.82 SLC6A4 (0.41) SLC6A4HRH3KDM4ESLC6A2SLC6A3
SCHEMBL10992363 0.82 SLC6A4 (0.45) SLC6A4HRH3SLC6A2UTS2R
SCHEMBL10991955 0.81 KDM4E (0.48) SLC6A4HRH3KDM4ESLC6A2SLC6A3
SCHEMBL10994963 0.81 SLC6A4 (0.35) SLC6A4HRH3KDM4EALDH1A1SLC6A2
SCHEMBL10994762 0.81 CHRNB2 (0.51) KDM4EFFAR1
SCHEMBL1919322 0.80 SLC6A2 (0.47) SLC6A4HRH3PPARGKDM4EPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4500541-A Pharmacologically active cyclopropane derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-02-19 US disclosed
EP-0039771-B1 CYCLOPROPANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PRODUCTION MERCK PATENT GmbH (DE) 1983-10-19 EP disclosed
EP-0039771-A1 Cyclopropane derivatives, pharmaceutical compositions containing them and processes for their production MERCK PATENT GmbH (DE) 1981-11-18 EP disclosed