SCHEMBL10985607

SCHEMBL10985607

CN(CCC(Oc1cccc(C(F)(F)F)c1)C1CC1)Cc1ccccc1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
KDM4E B2RXH2 1/20 0.58
SLC6A9 P48067 2/20 0.48
PPARG P37231 1/20 0.46
PPARA Q07869 1/20 0.46
LMNA P02545 1/20 0.44
HTT P42858 1/20 0.44
PAX8 Q06710 1/20 0.44
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TMEM97 Q5BJF2 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
DCUN1D1 Q96GG9 3/20 0.39
UBE2M P61081 2/20 0.39
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
FFAR1 O14842 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10989259 0.86 PPARG (0.43) ALDH1A1KDM4EPPARGPPARAMEN1
SCHEMBL10996291 0.85 SLC6A9 (0.44) ALDH1A1KDM4ESLC6A9PPARGPPARA
SCHEMBL10993880 0.85 CARM1 (0.44) LMNASIGMAR1
SCHEMBL10989374 0.84 SIGMAR1 (0.47) SIGMAR1OPRM1OPRL1
SCHEMBL10994633 0.84 ATM (0.40) ALDH1A1KDM4EMEN1KMT2ASIGMAR1
SCHEMBL10987323 0.84 GHSR (0.46) KDM4ETMEM97SIGMAR1
SCHEMBL10987479 0.84 TSHR (0.39) ALDH1A1KDM4ESIGMAR1
SCHEMBL10993995 0.84 KDM4E (0.40) ALDH1A1KDM4ESIGMAR1OPRM1
SCHEMBL10986644 0.82 TSHR (0.38) ALDH1A1KDM4ESIGMAR1DCUN1D1UBE2M
SCHEMBL12186131 0.81 SLC6A9 (0.70) ALDH1A1KDM4ESLC6A9PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4500541-A Pharmacologically active cyclopropane derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1985-02-19 US disclosed
EP-0039771-B1 CYCLOPROPANE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PRODUCTION MERCK PATENT GmbH (DE) 1983-10-19 EP disclosed
EP-0039771-A1 Cyclopropane derivatives, pharmaceutical compositions containing them and processes for their production MERCK PATENT GmbH (DE) 1981-11-18 EP disclosed