SCHEMBL10998617

SCHEMBL10998617

CC(=O)OC(SC(C)C)(c1ccccc1)c1ccncc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.42
CYP1A2 P05177 2/20 0.38
CYP2D6 P10635 1/20 0.38
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
EPHX2 P34913 1/20 0.35
CYP3A4 P08684 2/20 0.33
KCNN4 O15554 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
KCNH2 Q12809 1/20 0.33
ROCK2 O75116 1/20 0.33
RPS6KA5 O75582 1/20 0.33
MAP4K4 O95819 1/20 0.33
CDK1 P06493 1/20 0.33
CSF1R P07333 1/20 0.33
PRKACA P17612 1/20 0.33
FLT1 P17948 1/20 0.33
RPS6KB1 P23443 1/20 0.33
CDK2 P24941 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10992876 0.80 KIF11 (0.39) KIF11CYP2D6KMT2AMEN1CYP3A4
SCHEMBL10998615 0.79 KIF11 (0.42) KIF11CYP1A2CYP2D6KMT2AMEN1
SCHEMBL6535389 0.76 KCNN4 (0.42) KIF11CYP1A2CYP2D6KMT2AKCNN4
SCHEMBL10997363 0.73 KIF11 (0.42) KIF11CYP1A2CYP2D6KMT2AMEN1
Pyridine SCHEMBL8673561 0.69 CYP1A2 (0.39) KIF11CYP1A2CYP2D6KMT2AMEN1
SCHEMBL28320432 0.69 CYP19A1 (0.54) KIF11CYP17A1CYP19A1
SCHEMBL8695362 0.67 KIF11 (0.46) KIF11CYP1A2CYP2D6KMT2AMEN1
SCHEMBL10793742 0.67 ELANE (0.39) KIF11CYP1A2CYP2D6KMT2AMEN1
SCHEMBL4905934 0.67 ELANE (0.39) KIF11CYP1A2CYP2D6KMT2AMEN1
SCHEMBL10958637 0.67 ELANE (0.39) KIF11CYP1A2CYP2D6KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4535084-A ANTIARTHRITIC, ANTIINFLAMMATORY AGENTS PFIZER INC. (US) 1985-08-13 US disclosed
US-4246263-A ANTIARTHRITIC AGENTS PFIZER INC. (US) 1981-01-20 US disclosed