SCHEMBL11004012

SCHEMBL11004012

CCOC(=O)C1=C(C)N(C)C2=C(C(=O)OC2)C1c1cccc(Cl)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.50
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KDM4E B2RXH2 2/20 0.49
GAA P10253 1/20 0.49
ALDH1A1 P00352 2/20 0.48
POLB P06746 1/20 0.46
TSHR P16473 1/20 0.44
LMNA P02545 3/20 0.44
CACNA1F O60840 1/20 0.43
CACNA1D Q01668 1/20 0.43
CACNA1S Q13698 1/20 0.43
CACNA1C Q13936 1/20 0.43
ALOX12 P18054 2/20 0.42
HTT P42858 2/20 0.42
BCHE P06276 1/20 0.41
TP53 P04637 3/20 0.40
MDM2 Q00987 3/20 0.40
ADORA2B P29275 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11008812 0.91 GPBAR1 (0.42) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL9690849 0.85 KDM4E (0.39) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL11006883 0.79 KDM4E (0.77) HPGDKDM4EGAAALDH1A1CACNA1F
SCHEMBL8080875 0.75 ADORA2B (0.41) NPSR1HPGDSMN1; SMN2KDM4EALDH1A1
SCHEMBL11004817 0.75 KDM4E (0.47) NPSR1HPGDKDM4EGAAALDH1A1
SCHEMBL9865258 0.75 CYP3A4 (0.47) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL11007496 0.73 KDM4E (0.67) HPGDSMN1; SMN2KDM4EGAAALDH1A1
SCHEMBL11003915 0.72 KDM4E (0.45) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL11267200 0.72 NPSR1 (0.49) NPSR1HPGDSMN1; SMN2KDM4EGAA
SCHEMBL11003990 0.71 KDM4E (0.64) HPGDKDM4EGAAALDH1A1CACNA1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4532248-A Administering 1,4-dihydropyridine derivative exhibiting positive inotropic activity BAYER AKTIENGESELLSCHAFT (DE) 1985-07-30 US disclosed