SCHEMBL9690849

SCHEMBL9690849

CCOC(=O)OC1=C(C)N(C)C2=C(C(=O)OC2)C1c1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 2/20 0.39
MDM2 Q00987 7/20 0.39
TP53 P04637 6/20 0.39
CACNA1F O60840 1/20 0.38
CACNA1D Q01668 1/20 0.38
CACNA1S Q13698 1/20 0.38
CACNA1C Q13936 1/20 0.38
HPGD P15428 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 2/20 0.37
GLA P06280 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
HSD17B10 Q99714 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
BCHE P06276 1/20 0.36
POLB P06746 1/20 0.36
KDM1A O60341 1/20 0.35
RCOR1 Q9UKL0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11004012 0.85 NPSR1 (0.50) KDM4EALDH1A1MDM2TP53CACNA1F
SCHEMBL9689704 0.81 KDM4E (0.57) KDM4EALDH1A1MDM2TP53CACNA1F
SCHEMBL11008812 0.79 GPBAR1 (0.42) KDM4EALDH1A1HPGDNPSR1GAA
SCHEMBL10653759 0.77 CYP3A4 (0.39) KDM4EALDH1A1CACNA1CHPGDGAA
SCHEMBL9045462 0.77 SLC6A3 (0.38) NPSR1LMNA
SCHEMBL9691896 0.77 KDM4E (0.41) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL9691821 0.75 KDM4E (0.52) KDM4EALDH1A1MDM2TP53CACNA1F
SCHEMBL9691805 0.74 ALDH1A1 (0.36) KDM4EALDH1A1NPSR1GAASMN1; SMN2
SCHEMBL10817163 0.73 KDM4E (0.50) KDM4EALDH1A1CACNA1FCACNA1DCACNA1S
SCHEMBL11005887 0.73 CACNA1B (0.49) MDM2TP53CACNA1FCACNA1DCACNA1S

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed
EP-0071819-A1 Dihydropyridines with a positive inotropic activity, their use in pharmaceutical preparations, and processes for their preparation BAYER AG (DE) 1983-02-16 EP disclosed