SCHEMBL11005135

SCHEMBL11005135

CCc1nc2c(N)nc(-c3ccncc3)nc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
PRKCI P41743 5/20 0.36
ROCK2 O75116 5/20 0.35
GRK2 P25098 4/20 0.35
LATS1 O95835 2/20 0.35
LATS2 Q9NRM7 2/20 0.35
ADORA2A P29274 3/20 0.35
ADORA1 P30542 3/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ADORA3 P0DMS8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MAPK1 P28482 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11000644 0.81 GSK3B (0.40) PDE3BPDE3APRKCILATS1LATS2
SCHEMBL11004647 0.80 ADORA2A (0.39) PRKCILATS1LATS2ADORA2AADORA1
SCHEMBL14938324 0.78 LATS1 (0.34) PRKCIROCK2LATS1LATS2ADORA2A
SCHEMBL11005615 0.78 ADORA2A (0.33) PRKCIROCK2GRK2LATS1LATS2
SCHEMBL12006474 0.77 BMPR1B (0.42) NPC1ALDH1A1MAPTRAB9A
SCHEMBL11003505 0.77 GSK3B (0.43) PRKCILATS1LATS2ADORA2AADORA1
SCHEMBL11006980 0.77 MAPK14 (0.41) LATS1LATS2ADORA2AADORA1NPC1
SCHEMBL11005247 0.77 BRAF (0.41) PRKCIROCK2LATS1LATS2NPC1
SCHEMBL11004943 0.76 ALDH1A1 (0.41) LATS1LATS2ADORA2AADORA1NPC1
SCHEMBL12472696 0.75 ADORA2A (0.33) ADORA2AADORA1ALDH1A1MAPTADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4503228-A 2-(Pyridinyl)-4,5,6-pyrimidinetriamines STERLING DRUG INC. (US) 1985-03-05 US disclosed
US-4473571-A 8-Substituted-2-(4-pyridinyl)-9H-purin-6-amines and their cardiotonic use STERLING DRUG INC. (US) 1984-09-25 US disclosed