SCHEMBL11006162

SCHEMBL11006162

COc1cc(O)ccc1-c1nc2cncnc2[nH]1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 6/20 0.43
CCNA2 P20248 6/20 0.43
CCND1 P24385 6/20 0.43
CDK2 P24941 6/20 0.43
CCND3 P30281 6/20 0.43
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
PDE5A O76074 3/20 0.41
PDE3B Q13370 1/20 0.41
PDE3A Q14432 1/20 0.41
CHEK1 O14757 1/20 0.41
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
KDR P35968 1/20 0.41
JAK3 P52333 1/20 0.41
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
LCK P06239 1/20 0.38
FGFR1 P11362 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11011297 0.86 IMPDH2 (0.45) PDE5APDE3BPDE3APDE2A
SCHEMBL11237399 0.86 PDE2A (0.51) PDE5APDE3BPDE3AKMT2AGAA
SCHEMBL11356780 0.85 AMY1A (0.47) PDE5APDE3BPDE3A
SCHEMBL10689035 0.82 ESR1 (0.42) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL10962015 0.82 ESR1 (0.36) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL4839233 0.81 ESR1 (0.41) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL11237474 0.81 CYP17A1 (0.42) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL11228926 0.81 PDE5A (0.38) PDE5APDE3BPDE3AKMT2APDE2A
SCHEMBL10869538 0.81 SLC2A1 (0.44) PDE5APDGFRBPDGFRAKMT2AGAA
SCHEMBL10749457 0.80 PDE2A (0.50) CDK4CCNA2CCND1CDK2CCND3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142075-A2 Purine derivatives, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-05-22 EP disclosed