SCHEMBL10962015

SCHEMBL10962015

COc1c(-c2nc3cncnc3[nH]2)ccc2cc(O)ccc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 2/20 0.36
ESR2 Q92731 2/20 0.36
CDK4 P11802 3/20 0.36
CDK2 P24941 3/20 0.36
CCNA2 P20248 2/20 0.36
CCND1 P24385 2/20 0.36
CCND3 P30281 2/20 0.36
AMY1A P0DUB6 4/20 0.35
AURKA O14965 1/20 0.35
CDK1 P06493 1/20 0.35
AURKB Q96GD4 1/20 0.35
CYP17A1 P05093 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP11B1 P15538 2/20 0.34
CYP11B2 P19099 2/20 0.34
FTO Q9C0B1 1/20 0.34
CHEK1 O14757 1/20 0.34
JAK2 O60674 1/20 0.34
JAK1 P23458 1/20 0.34
TYK2 P29597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10960693 0.84 EGFR (0.36) AMY1ACYP17A1CYP3A4CYP11B1CYP11B2
SCHEMBL11006162 0.82 CDK4 (0.43) ESR1ESR2CDK4CDK2CCNA2
SCHEMBL10962019 0.82 GUSB (0.40) ESR1ESR2CDK4CDK2CCNA2
SCHEMBL10965537 0.80 EGFR (0.44) AMY1ACYP17A1CYP3A4CYP11B1CYP11B2
SCHEMBL10963776 0.79 PDE5A (0.39) AMY1ACDK1CYP3A4
SCHEMBL10965860 0.78 EGFR (0.32) AMY1AEGFR
SCHEMBL11233385 0.75 AMY1A (0.41) AMY1ACYP3A4EGFR
SCHEMBL10960260 0.73 ALDH1A1 (0.35) EGFRLMNA
SCHEMBL10983982 0.72 CYP17A1 (0.33) AMY1ACYP17A1CYP11B1CYP11B2EGFR
SCHEMBL10959064 0.72 MAPT (0.30) KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0142235-A1 Naphthalenylimidazopyridine and derivatives and their preparation ELI LILLY AND COMPANY (US) 1985-05-22 EP disclosed
US-4515796-A INOTROPIC, BRONCHODILATOR, VASODILATORS, ANTICOAGULANTS ELI LILLY AND COMPANY (US) 1985-05-07 US disclosed