SCHEMBL11007804

SCHEMBL11007804

CCOC(=O)C1=C(N)NC(C)=CC1c1ccccc1Cl

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.54
POLB P06746 1/20 0.54
CACNA1D Q01668 5/20 0.50
CYP2C9 P11712 4/20 0.50
CYP3A4 P08684 3/20 0.50
CYP2C19 P33261 3/20 0.50
TBXA2R P21731 3/20 0.50
ADRA1A P35348 3/20 0.50
SLC6A3 Q01959 3/20 0.50
CACNA1C Q13936 3/20 0.50
KDM4E B2RXH2 2/20 0.50
MEN1 O00255 2/20 0.50
CYP1A2 P05177 2/20 0.50
KMT2A Q03164 2/20 0.50
HIF1A Q16665 2/20 0.50
HSD17B10 Q99714 2/20 0.50
ALDH1A1 P00352 2/20 0.50
LMNA P02545 2/20 0.50
ABCB11 O95342 2/20 0.50
ABCB1 P08183 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11803207 0.89 CA1 (0.50) TSHRPOLBCACNA1DCYP2C9CYP3A4
SCHEMBL11795742 0.86 CACNA1D (0.58) TSHRPOLBCACNA1DCYP2C9CYP3A4
SCHEMBL9689480 0.84 TSHR (0.43) TSHRPOLBCACNA1DCYP2C9CYP3A4
SCHEMBL11793306 0.84 ALOX15 (0.54) KDM4EHSD17B10ALDH1A1HPGDGAA
SCHEMBL11799255 0.83 CACNA1D (0.60) CACNA1DKDM4EALDH1A1ADORA3GAA
SCHEMBL14297933 0.81 TBXA2R (0.67) TSHRPOLBCACNA1DCYP2C9CYP3A4
SCHEMBL11800413 0.80 CACNA1D (0.51) CACNA1DCYP2C9CYP3A4CYP2C19CACNA1C
SCHEMBL11523639 0.80 CYP2C9 (0.65) TSHRPOLBCACNA1DCYP2C9CYP3A4
SCHEMBL3017208 0.78 CYP2C9 (0.73) TSHRPOLBCACNA1DCYP2C9CYP3A4
SCHEMBL11524317 0.76 KDM4E (0.73) TSHRPOLBCACNA1DCYP2C9CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4532248-A Administering 1,4-dihydropyridine derivative exhibiting positive inotropic activity BAYER AKTIENGESELLSCHAFT (DE) 1985-07-30 US disclosed
US-3989708-A HYPOTENSIVE, CORONARY VESSEL DILATORS BAYER AKTIENGESELLSCHAFT (DT) 1976-11-02 US disclosed