SCHEMBL11008652

SCHEMBL11008652

COc1ccc2c(c1)CCC(NCC(=O)O)C2

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACHE P22303 5/20 0.62
CA1 P00915 4/20 0.62
CA2 P00918 4/20 0.62
DRD2 P14416 4/20 0.60
DRD3 P35462 4/20 0.60
MTNR1A P48039 2/20 0.60
MTNR1B P49286 1/20 0.60
CYP26A1 O43174 1/20 0.51
GRIN1 Q05586 1/20 0.51
GRIN2B Q13224 1/20 0.51
POLB P06746 1/20 0.48
KMT2A Q03164 1/20 0.48
CYP19A1 P11511 1/20 0.48
HTR1D P28221 1/20 0.46
ADRB1 P08588 1/20 0.45
ADRB3 P13945 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11009077 0.95 DRD2 (0.67) ACHECA1CA2DRD2DRD3
SCHEMBL11005303 0.85 DRD2 (0.58) ACHECA1CA2DRD2DRD3
Hydrochloric Acid SCHEMBL11005295 0.84 DRD2 (0.57) ACHECA1CA2DRD2DRD3
SCHEMBL10765415 0.82 DRD2 (0.71) ACHECA1CA2DRD2DRD3
SCHEMBL11493562 0.82 DRD2 (0.71) ACHECA1CA2DRD2DRD3
SCHEMBL18983605 0.81 CA1 (0.58) ACHECA1CA2DRD2DRD3
Hydrochloric Acid SCHEMBL11443133 0.81 DRD2 (0.69) ACHECA1CA2DRD2DRD3
SCHEMBL11007069 0.81 DRD2 (0.65) ACHECA1CA2DRD2DRD3
SCHEMBL607070 0.80 DRD2 (0.90) ACHECA1CA2DRD2DRD3
SCHEMBL3975748 0.80 MTNR1A (0.90) ACHECA1CA2DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4521607-A HYPOTENSIVE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1985-06-04 US disclosed
EP-0035868-A1 Bicyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1981-09-16 EP disclosed