SCHEMBL11014615

SCHEMBL11014615

COc1ccc2nc3sc(C(=O)O)cn3c(=O)c2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALPG P10696 1/20 0.60
KDM4E B2RXH2 5/20 0.47
HSD17B10 Q99714 4/20 0.47
ALDH1A1 P00352 4/20 0.47
HPGD P15428 4/20 0.47
POLB P06746 1/20 0.47
LMNA P02545 2/20 0.44
PLA2G2A P14555 3/20 0.43
TSHR P16473 2/20 0.41
USP2 O75604 1/20 0.41
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.41
TBXAS1 P24557 1/20 0.40
PTAFR P25105 1/20 0.40
DHODH Q02127 1/20 0.40
ATM Q13315 1/20 0.40
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9770670 0.93 ALPG (0.55) ALPGKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL11249330 0.83 ALPG (0.55) ALPGKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL29660149 0.82 SMN1; SMN2 (0.48) ALPGKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL18548584 0.82 SMN1; SMN2 (0.48) ALPGKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL10696645 0.81 ALPG (0.53) ALPGKDM4EHSD17B10ALDH1A1HPGD
SCHEMBL11014908 0.80 DHODH (0.40) ALPGMAPTDHODHMEN1KMT2A
SCHEMBL11015093 0.80 PTAFR (0.42) TBXAS1PTAFR
SCHEMBL10848968 0.78 TXNRD1 (0.47) ALPGKDM4EALDH1A1HPGDMAPT
SCHEMBL11015097 0.78 MEN1 (0.39) ALPGKDM4EALDH1A1HPGDPOLB
SCHEMBL11018500 0.78 ALPG (0.37) ALPGMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0006114-B1 7-METHOXY-5-OXO-5H-THIAZOLO(2,3-B)QUINAZOLIN-2-CARBOXYLIC ACID AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1982-04-07 EP claimed
US-4168380-A ANTIALLERGEN HOFFMANN-LA ROCHE INC. (US) 1979-09-18 US claimed
EP-0142057-A2 Thiazoloquinazoline derivatives, their preparation and pharmaceutical compositions containing same F. HOFFMANN-LA ROCHE AG (CH) 1985-05-22 EP disclosed
US-4282360-A ANTIALLERGENS HOFFMANN-LA ROCHE INC. (US) 1981-08-04 US disclosed
EP-0006114-A1 7-Methoxy-5-oxo-5H-thiazolo(2,3-b)quinazolin-2-carboxylic acid and its pharmaceutically acceptable salts, process for their preparation and medicines containing them F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft (CH) 1980-01-09 EP disclosed
US-4168380-A ANTIALLERGEN HOFFMANN-LA ROCHE INC. (US) 1979-09-18 US disclosed
US-4168380-A ANTIALLERGEN HOFFMANN-LA ROCHE INC. (US) 1979-09-18 US disclosed
US-4168380-A ANTIALLERGEN HOFFMANN-LA ROCHE INC. (US) 1979-09-18 US disclosed