SCHEMBL11016276

SCHEMBL11016276

Nc1nc(=O)n(CC2CC2)c(=O)[nH]1

nearest known ligand 0.54

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 6/20 0.54
PDE4A P27815 6/20 0.54
PDE4B Q07343 6/20 0.54
PDE4C Q08493 6/20 0.54
PDE4D Q08499 6/20 0.54
MEN1 O00255 1/20 0.53
ALDH1A1 P00352 1/20 0.53
CYP3A4 P08684 1/20 0.53
KMT2A Q03164 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
MTOR P42345 3/20 0.38
GRIN1 Q05586 2/20 0.37
GRIN2B Q13224 2/20 0.37
TLR7 Q9NYK1 7/20 0.37
TLR8 Q9NR97 4/20 0.37
MAP3K11 Q16584 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23202302 0.76 PDE5A (0.48) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7345942 0.76 PDE5A (0.62) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL7345938 0.76 PDE5A (0.66) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL27164821 0.73 PNP (0.32) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL27164823 0.71 HSD17B10 (0.41) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL11036035 0.70 ALDH1A1 (0.40) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL1546788 0.70 ALDH1A1 (0.54) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL26907658 0.70 XDH (0.32) SMN1; SMN2TLR7
SCHEMBL1943792 0.70 ALDH1A1 (0.54) PDE5APDE4APDE4BPDE4CPDE4D
Cipamfylline SCHEMBL26990 0.70 PDE4A (1.00) PDE5APDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0154906-A2 3-Cyclopropylmethyl-1,3,5-triazine-2,4-dione BAYER AG (DE) 1985-09-18 EP claimed