SCHEMBL1101690

SCHEMBL1101690

COc1ccc2c(O[C@@H]3C[C@@H](C(=O)O)N(C(=O)CC(C)(C)C)C3)cc(-c3nc(C(C)C)cs3)nc2c1C

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.43
CTSB P07858 1/20 0.37
PPP3CB P16298 1/20 0.37
ADRB3 P13945 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
ABCC1 P33527 1/20 0.32
ABCC2 Q92887 1/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
ERBB2 P04626 2/20 0.32
SLC5A7 Q9GZV3 1/20 0.30
AGTR2 P50052 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1101687 0.94 CTSS (0.44) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL7936436 0.89 CTSS (0.44) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL1101734 0.89 CTSS (0.44) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL13337167 0.87 CTSS (0.48) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL1101688 0.83 CTSS (0.44) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL883040 0.83 CTSS (0.43) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL12775112 0.82 UCHL1 (0.38) CTSSCTSBPPP3CBADRB3ADRA2B
SCHEMBL14353637 0.82 CTSS (0.49) CTSSADRB3ADRA2BADRA2CSLC5A7
SCHEMBL313204 0.82 UCHL1 (0.38) CTSSCTSBPPP3CBABCC1ABCC2
SCHEMBL2213932 0.82 UCHL1 (0.38) CTSSCTSBPPP3CBABCC1ABCC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153800-B2 Macrocyclic inhibitors of hepatitis C virus TIBOTEC PHARMACEUTICALS LTD. (IE) 2012-04-10 US disclosed
US-8153800-B2 Macrocyclic inhibitors of hepatitis C virus TIBOTEC PHARMACEUTICALS LTD. (IE) 2012-04-10 US disclosed