SCHEMBL11018705

SCHEMBL11018705

COc1cc(SCC#N)ccc1-c1nc2cc(F)ccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 15/20 0.47
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
PDE10A Q9Y233 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDE5A O76074 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9634871 0.83 PDE5A (0.47) AMY1AKDM4EALDH1A1TP53PDE10A
SCHEMBL10742496 0.83 PDE5A (0.43) AMY1AKDM4EALDH1A1TP53PDE10A
SCHEMBL11019179 0.80 AMY1A (0.47) AMY1APDE5A
SCHEMBL10762222 0.78 AMY1A (0.41) AMY1AKDM4EALDH1A1NPC1SMN1; SMN2
SCHEMBL11017329 0.76 AR (0.50) AMY1AKDM4EALDH1A1TP53SMN1; SMN2
SCHEMBL11009297 0.76 PDE5A (0.35) AMY1AKDM4EALDH1A1TP53PDE10A
SCHEMBL10748409 0.76 AMY1A (0.56) AMY1A
SCHEMBL10737588 0.74 PDE2A (0.42) KDM4EALDH1A1TP53PDE10APDE5A
SCHEMBL10760601 0.74 MAPK10 (0.42) AMY1ANPC1RAB9APDE5A
SCHEMBL9635715 0.73 PDE5A (0.47) AMY1AKDM4EALDH1A1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed