SCHEMBL10762222

SCHEMBL10762222

CCSc1ccc(-c2nc3cc(C#N)ccc3[nH]2)c(OC)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 7/20 0.41
MAPK10 P53779 1/20 0.41
AR P10275 3/20 0.39
F7 P08709 1/20 0.37
PDE5A O76074 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2C19 P33261 2/20 0.36
PKN1 Q16512 1/20 0.36
PKN2 Q16513 1/20 0.36
RHEB Q15382 1/20 0.36
CYP2E1 P05181 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C8 P10632 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2B6 P20813 1/20 0.36
KDM4E B2RXH2 2/20 0.35
ALDH1A1 P00352 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11017329 0.92 AR (0.50) AMY1AMAPK10ARF7PDE5A
SCHEMBL11018943 0.92 AMY1A (0.47) AMY1AF7CYP1A2CYP2C9CYP2C19
SCHEMBL10760601 0.88 MAPK10 (0.42) AMY1AMAPK10PDE5APDE3BPDE3A
SCHEMBL11017363 0.83 AR (0.50) AMY1AARF7CYP1A2CYP2C9
SCHEMBL10765326 0.81 MAPK10 (0.42) AMY1AMAPK10F7PDE5APKN1
SCHEMBL10748660 0.81 CDK4 (0.46) AMY1AMAPK10F7PDE5APDE3B
SCHEMBL11021670 0.81 PDE5A (0.38) MAPK10PDE5ACYP1A2CYP2C9CYP2C19
SCHEMBL11017897 0.80 PDE4A (0.44) AMY1ANPC1MAPT
SCHEMBL10763275 0.80 MAPK10 (0.42) MAPK10PDE5APDE3BPDE3ACYP1A2
SCHEMBL11016458 0.79 CHEK2 (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0209707-A2 2-Aryl imidazoles, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1987-01-28 EP disclosed
EP-0148431-A1 Benzimidazoles, their preparation, and medicaments containing these compounds Dr. Karl Thomae GmbH (DE) 1985-07-17 EP disclosed