SCHEMBL11021076

SCHEMBL11021076

CC1CC1c1[nH]c2c(F)c(F)c(F)cc2c(=O)c1C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 2/20 0.32
GSK3A P49840 2/20 0.32
GSK3B P49841 2/20 0.32
PIM3 Q86V86 2/20 0.32
PRKD3 O94806 1/20 0.32
IRAK1 P51617 1/20 0.32
RPS6KA3 P51812 1/20 0.32
DYRK1A Q13627 1/20 0.32
CSNK1G3 Q9Y6M4 1/20 0.32
CSNK1G1 Q9HCP0 1/20 0.32
KCNH2 Q12809 1/20 0.32
CAT P04040 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11020992 0.80 PIM1 (0.56) PIM1GSK3AGSK3BPIM3PRKD3
SCHEMBL10911793 0.74 KCNH2 (0.41) KCNH2ALDH1A1
SCHEMBL9877122 0.74 KCNH2 (0.36) KCNH2KDM4EALDH1A1HPGDHSD17B10
SCHEMBL10950502 0.74 EIF4A3 (0.39) KCNH2
SCHEMBL11020858 0.73 KCNH2 (0.32) KCNH2KDM4EALDH1A1
SCHEMBL6004835 0.72 POLB (0.34) PIM1GSK3AGSK3BPIM3CSNK1G1
SCHEMBL6904311 0.70 KMT2A (0.39) KDM4EALDH1A1HPGD
SCHEMBL16098745 0.67 TOP2A (0.50) KCNH2
SCHEMBL6341275 0.67 HCAR2 (0.35) PIM1GSK3AGSK3BPIM3PRKD3
SCHEMBL3802263 0.66 PRKAB2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0153163-A2 7-Substituted-1-cyclopropyl-6,8-difluoro-1,4-dihydro-4-oxo-3-quinolinecarboxylic acids; 7-substituted-1-cyclopropyl-1,4-dihydro-6-fluoro-4-oxo-1,8-naphthyridine-3-carboxylic acids; their derivatives; and a process for preparing the compounds WARNER-LAMBERT COMPANY (US) 1985-08-28 EP disclosed