SCHEMBL16098745

SCHEMBL16098745

O=C(O)c1c(C2CC2)[nH]c2c(F)c(-c3ccncc3)c(F)cc2c1=O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 9/20 0.50
TOP2B Q02880 9/20 0.50
CDC7 O00311 2/20 0.35
MAPK11 Q15759 2/20 0.34
MAPK14 Q16539 2/20 0.34
KCNH2 Q12809 1/20 0.34
PRKAB2 O43741 1/20 0.32
PRKAG1 P54619 1/20 0.32
PRKAA2 P54646 1/20 0.32
PRKAA1 Q13131 1/20 0.32
PRKAG3 Q9UGI9 1/20 0.32
PRKAG2 Q9UGJ0 1/20 0.32
PRKAB1 Q9Y478 1/20 0.32
HCAR2 Q8TDS4 1/20 0.32
FABP4 P15090 1/20 0.32
FABP5 Q01469 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004835 0.76 POLB (0.34) HCAR2
SCHEMBL6341275 0.74 HCAR2 (0.35) TOP2ATOP2BHCAR2
SCHEMBL6904417 0.70 IDO1 (0.38) KCNH2PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL11021076 0.67 PIM1 (0.32) KCNH2
SCHEMBL6904311 0.67 KMT2A (0.39)
SCHEMBL7557799 0.67 ALDH1A1 (0.51) TOP2ATOP2B
SCHEMBL16121059 0.67 TOP2A (1.00) TOP2ATOP2B
SCHEMBL8061645 0.66 DPP4 (0.39)
SCHEMBL4237180 0.65 PADI4 (0.36) HCAR2
SCHEMBL10738605 0.65 TOP2A (0.52) TOP2ATOP2BCDC7MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014152895-A1 MULTI-TIERED HIGH THROUGH-PUT SCREEN FOR COMPOUNDS EFFECTIVE AGAINST BACTERIAL BIOFILM AND COMPOUNDS EFFECTIVE FOR INHIBITING AND ERADICATING BACTERIAL BIOFILM UNIVERSITY OF CINCINNATI (US) 2014-09-25 WO disclosed