SCHEMBL11022689

SCHEMBL11022689

CCCCC(CCC(CCc1ccccc1)NC)(CN(C)C)c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SIGMAR1 Q99720 6/20 0.35
EBP Q15125 3/20 0.35
MMP2 P08253 3/20 0.35
MMP3 P08254 3/20 0.35
SLC6A2 P23975 2/20 0.32
SLC6A4 P31645 2/20 0.32
SLC6A3 Q01959 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
KCNH2 Q12809 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11022708 0.79 TAAR1 (0.36) SIGMAR1EBPMMP2MMP3
SCHEMBL11022683 0.78 SIGMAR1 (0.49) SIGMAR1KCNH2
SCHEMBL11022687 0.77 SIGMAR1 (0.58) SIGMAR1EBPSLC6A2SLC6A4SLC6A3
SCHEMBL22117248 0.75 SIGMAR1 (0.47) CYP1A2CYP2C9CYP2C19SIGMAR1MMP2
SCHEMBL11022228 0.74 SIGMAR1 (0.50) SIGMAR1EBPKCNH2
SCHEMBL11022231 0.72 SIGMAR1 (0.65) SIGMAR1EBPKCNH2
SCHEMBL27999740 0.72 SIGMAR1 (0.53) SIGMAR1SLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL11024418 0.71 KCNH2 (0.35) SIGMAR1EBPSLC6A2SLC6A4SLC6A3
SCHEMBL6560515 0.70 KIF11 (0.42) SIGMAR1
SCHEMBL13061188 0.69 TAAR1 (0.47) SIGMAR1SLC6A2SLC6A4SLC6A3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0082266-B1 SUBSTITUTED 1,5-DIAMINOPENTANES, THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BASF Aktiengesellschaft (DE) 1985-01-09 EP disclosed
EP-0082266-A1 Substituted 1,5-diaminopentanes, their preparation and pharmaceutical compositions containing them BASF Aktiengesellschaft (DE) 1983-06-29 EP disclosed