SCHEMBL11023760

SCHEMBL11023760

CC(O)N(c1nc(N2CC[S+]([O-])CC2)c2ncnc(OCc3ccc(F)cc3)c2n1)C(C)O

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KIT P10721 1/20 0.34
ACACB O00763 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
DAPK1 P53355 1/20 0.32
HRH4 Q9H3N8 1/20 0.30
CSNK1A1 P48729 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11026806 0.92 HRH4 (0.38) KITALDH1A1LMNAHPGDTSHR
SCHEMBL11028075 0.91 HRH4 (0.39) ALDH1A1LMNAHPGDTSHRMAPK1
SCHEMBL11026793 0.91 ALDH1A1 (0.43) KITALDH1A1LMNAHPGDTSHR
SCHEMBL11044328 0.90 HRH4 (0.40) KITALDH1A1LMNAHPGDTSHR
SCHEMBL11312367 0.90 ACACB (0.35) KITACACBALDH1A1LMNAHPGD
SCHEMBL11026067 0.87 NPC1 (0.31) ALDH1A1HRH4
SCHEMBL11029550 0.86 PDGFRB (0.34) KITALDH1A1TSHRHTT
SCHEMBL11046483 0.86 ACACB (0.34) ACACBCSNK1A1
SCHEMBL11047615 0.85 HRH4 (0.40) ACACBALDH1A1LMNAHPGDTSHR
SCHEMBL11028231 0.85 PDE5A (0.43) KITALDH1A1LMNAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055444-B1 TRISUBSTITUTED PYRIMIDO(5,4-D)PYRIMIDINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1985-03-20 EP disclosed