SCHEMBL11029550

SCHEMBL11029550

COc1ccc(COc2ncnc3c(N4CC[S+]([O-])CC4)nc(N(C(C)O)C(C)O)nc23)cc1OC

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 3/20 0.34
PDGFRA P16234 2/20 0.34
PI4KB Q9UBF8 1/20 0.34
KIT P10721 5/20 0.33
PDE5A O76074 1/20 0.33
TLR9 Q9NR96 4/20 0.33
TLR7 Q9NYK1 4/20 0.33
TSHR P16473 1/20 0.33
HTT P42858 1/20 0.33
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
HSD17B10 Q99714 1/20 0.32
STAT3 P40763 1/20 0.31
GAK O14976 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11044328 0.89 HRH4 (0.40) KITPDE5ATSHRHTTALDH1A1
SCHEMBL11026067 0.87 NPC1 (0.31) ALDH1A1
SCHEMBL11026806 0.87 HRH4 (0.38) KITTSHRHTTALDH1A1
SCHEMBL11046232 0.86 BCHE (0.33) KITTSHRHTTALDH1A1KDM4E
SCHEMBL11028075 0.86 HRH4 (0.39) TSHRHTTALDH1A1
SCHEMBL11023760 0.86 KIT (0.34) KITTSHRHTTALDH1A1
SCHEMBL11026793 0.86 ALDH1A1 (0.43) KITTLR9TLR7TSHRHTT
SCHEMBL11025913 0.85 SLC29A1 (0.33) PDE5ATSHRALDH1A1KDM4EHSD17B10
SCHEMBL11028231 0.85 PDE5A (0.43) PDGFRBPDGFRAKITPDE5ATSHR
SCHEMBL11312367 0.85 ACACB (0.35) KITTSHRHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055444-B1 TRISUBSTITUTED PYRIMIDO(5,4-D)PYRIMIDINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1985-03-20 EP disclosed
US-4478833-A ANTICOAGULANTS DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-10-23 US disclosed
EP-0055444-A2 Trisubstituted pyrimido(5,4-d)pyrimidines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-07-07 EP disclosed