SCHEMBL11028075

SCHEMBL11028075

CC(O)N(c1nc(N2CC[S+]([O-])CC2)c2ncnc(OCc3ccc(Cl)cc3)c2n1)C(C)O

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 5/20 0.39
LMNA P02545 2/20 0.33
HTT P42858 2/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
DAPK1 P53355 1/20 0.32
PDE10A Q9Y233 1/20 0.31
ACHE P22303 1/20 0.30
BACE1 P56817 1/20 0.30
AKT1 P31749 1/20 0.30
AKT2 P31751 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11026806 0.92 HRH4 (0.38) HRH4LMNAHTTALDH1A1HPGD
SCHEMBL11023760 0.91 KIT (0.34) HRH4LMNAHTTALDH1A1HPGD
SCHEMBL11026793 0.91 ALDH1A1 (0.43) HRH4LMNAHTTALDH1A1HPGD
SCHEMBL11026067 0.90 NPC1 (0.31) HRH4ALDH1A1AKT1AKT2
SCHEMBL11044328 0.90 HRH4 (0.40) HRH4LMNAHTTALDH1A1HPGD
SCHEMBL11021816 0.88 MEN1 (0.32) HTTALDH1A1AKT1AKT2
SCHEMBL11031948 0.86 CSF1R (0.32) ALDH1A1HPGDTSHR
SCHEMBL11029550 0.86 PDGFRB (0.34) HTTALDH1A1TSHR
SCHEMBL11026550 0.86 CNR2 (0.33) LMNAALDH1A1HPGDAKT1AKT2
SCHEMBL11028231 0.85 PDE5A (0.43) LMNAHTTALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0055444-B1 TRISUBSTITUTED PYRIMIDO(5,4-D)PYRIMIDINES, THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1985-03-20 EP disclosed
US-4478833-A ANTICOAGULANTS DR. KARL THOMAE GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1984-10-23 US disclosed
EP-0055444-A2 Trisubstituted pyrimido(5,4-d)pyrimidines, their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1982-07-07 EP disclosed